H2L 5765834

CAS No. 420841-84-5

H2L 5765834( —— )

Catalog No. M24386 CAS No. 420841-84-5

H2L 5765834 is a lysophosphatidic acid receptors antagonist.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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5MG 110 In Stock
10MG 177 In Stock
25MG 410 In Stock
50MG 605 In Stock
100MG 860 In Stock
500MG 1728 In Stock
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Biological Information

  • Product Name
    H2L 5765834
  • Note
    Research use only, not for human use.
  • Brief Description
    H2L 5765834 is a lysophosphatidic acid receptors antagonist.
  • Description
    H2L 5765834 is a lysophosphatidic acid receptors antagonist.
  • In Vitro
    H2L 5765834 displays no effect on LPA2 or LPA4 receptors.H2L 5765834 inhibits LPA-induced platelet shape change with an IC50 of 13.73±2.52 μM.
  • In Vivo
    H2L 5765834 (20 mg/kg; i.p.) could not affect the LPA-induced decrease of alanine transaminase (ALT) in the acetaminophen (APAP) overdose-induced acute liver injury model.
  • Synonyms
    ——
  • Pathway
    GPCR/G Protein
  • Target
    LPA Receptor
  • Recptor
    lysophosphatidic acid receptors
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    420841-84-5
  • Formula Weight
    404.33
  • Molecular Formula
    C21H12N2O7
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO:40mg/ml(98.93mM; need ultrasonic)
  • SMILES
    [O-][N+](c(cc1)ccc1Oc1cc(N(C(c(cc2)c3cc2C(O)=O)=O)C3=O)ccc1)=O
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

molnova catalog
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